BDBM50260093 CHEMBL4078100

SMILES COc1nnc2ccc(nn12)N1CCC(CC1)c1ccc(OCCN2CCN(C)C(=O)[C@H]2C)cc1

InChI Key InChIKey=RSMYFSPOTCDHHJ-GOSISDBHSA-N

Data  17 KI  10 IC50

PDB links: 1 PDB ID matches this monomer.

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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50260093   

TargetHistone acetyltransferase p300(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50260093(CHEMBL4078100)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human EP300 expressed in bacterial expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed